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Discovery of imidazo[1,2-a]-, [1,2,4]triazolo[4,3-a]-, and [1,2,4]triazolo[1,5-a]pyridine-8-carboxamide negative allosteric modulators of metabotropic glutamate receptor subtype 5
| Content Provider | Scilit |
|---|---|
| Author | Felts, Andrew S. Rodriguez, Alice L. Morrison, Ryan D. Bollinger, Katrina A. Venable, Daryl F. Blobaum, Anna L. Byers, Frank W. Gray, Analisa Thompson Daniels, J. Scott Niswender, Colleen M. Jones, Carrie K. Conn, P. Jeffrey Lindsley, Craig W. Emmitte, Kyle A. |
| Copyright Year | 2017 |
| Description | Journal: Bioorganic & medicinal chemistry letters |
| Related Links | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5716465/pdf |
| Ending Page | 4866 |
| Page Count | 9 |
| Starting Page | 4858 |
| ISSN | 0960894X |
| DOI | 10.1016/j.bmcl.2017.09.042 |
| Journal | Bioorganic & medicinal chemistry letters |
| Issue Number | 21 |
| Volume Number | 27 |
| Language | English |
| Publisher | Elsevier BV |
| Publisher Date | 2017-11-01 |
| Access Restriction | Open |
| Subject Keyword | Journal: Bioorganic & medicinal chemistry letters Medicinal Chemistry Metabotropic Glutamate Receptor Subtype 5 (mglu5) Negative Allosteric Modulator (nam) Central Nervous System (cns) G-protein Coupled Receptor (gpcr) |
| Content Type | Text |
| Resource Type | Article |
| Subject | Organic Chemistry Drug Discovery Biochemistry Molecular Biology Clinical Biochemistry Molecular Medicine Pharmaceutical Science |