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Enhancing Drug Residence Time by Shielding of Intra-Protein Hydrogen Bonds: A Case Study on CCR2 Antagonists
| Content Provider | Scilit |
|---|---|
| Author | Magarkar, Aniket Schnapp, Gisela Apel, Anna-Katharina Seeliger, Daniel Tautermann, Christofer S. |
| Copyright Year | 2019 |
| Related Links | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6421533/pdf |
| Ending Page | 328 |
| Page Count | 5 |
| Starting Page | 324 |
| ISSN | 19485875 |
| e-ISSN | 19485875 |
| DOI | 10.1021/acsmedchemlett.8b00590 |
| Journal | ACS Medicinal Chemistry Letters |
| Issue Number | 3 |
| Volume Number | 10 |
| Language | English |
| Publisher | American Chemical Society (ACS) |
| Publisher Date | 2019-03-14 |
| Access Restriction | Open |
| Subject Keyword | Journal: ACS Medicinal Chemistry Letters Medicinal Chemistry Water Networks Drug Residence Time Buried Hydrogen Bonds |
| Content Type | Text |
| Resource Type | Article |
| Subject | Organic Chemistry Drug Discovery Biochemistry |